enquiry@advinus.eurofinsasia.com

Journal Article/Patents

Functional observational battery (FOB) tests using caffeine and chlorpromazine hydrochloride in sprague-dawley rats” Subramanian Baskaran,Prakash Malaiarasan,Sanjaykumar Mansukhlal Paneliya. Cellular and Molecular Biology (8 October 2024), 70(9), DOI:10.14715/cmb/2024.70.9.2

A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties” Antonio Laghezza, Carmen Cerchia, Massimo Genovese, Roberta Montanari, Davide Capelli, Judith Wackerlig, Stefan Simic, Emanuele Falbo, Lucia Pecora, Rosalba Leuci, Leonardo Brunetti, Luca Piemontese, Paolo Tortorella, Abanish Biswas, Ravi Pratap Singh, Suhas Tambe, C.A. Sudeep, Ashok Kumar Pattnaik, Venkatesan Jayaprakash, Paolo Paoli, Antonio Lavecchia, Fulvio Loiodice. Science Direct (5 September 2024), 275, DOI:10.1016/j.ejmech.2024.116567

Carbohydrate fatty acid monosulphate ester is a potent adjuvant for low-dose seasonal influenza vaccines” Peter Paul L.I. Platenburg, Frantz Deschamps, Jennifer Jung, Clément Leonard, Séverine Rusconi, S.B. Mohan Kumar, S.M. Sulaiman, Leon de Waal, Luuk A. Th. Hilgers. Science Direct (31 October 2023), DOI:10.1016/j.vaccine.2023.10.017

Analysis of Quinolinequinone Analogs with Promising Cytotoxic Activity against Breast Cancer” Ayse Mine Yilmaz Goler, Ayse Tarbin Jannuzzi, Abanish Biswas, Subodh Mondal, Vinay N Basavanakatti, Raghusrinivasan Jayaprakash Venkatesan, Hatice Yıldırım, Mahmut Yıldız, Hülya Çelik Onar, Nilüfer Bayrak, Venkatesan Jayaprakash, Amaç Fatih TuYuN. (23 August 2023), DOI:10.1002/cbdv.202300848

Cytotoxic activity of quinolinequinones in cancer: In vitro studies, molecular docking, and ADME/PK profiling” Ayse Tarbin Jannuzzi, Ayse Mine Yilmaz Goler, Deepak Shilkar, Subodh Mondal, Vinay N. Basavanakatti, Hatice Yıldırım, Mahmut Yıldız, Hülya Çelik Onar, Nilüfer Bayrak, Venkatesan Jayaprakash, Amaç Fatih TuYuN. Wiley Online Library (03 August 2023), DOI:10.1111/cbdd.14314

Pregnancy-associated Steroid Effects on Insulin Sensitivity, Adipogenesis, and Lipogenesis: Role of Wnt/β-Catenin Pathway” Neethu Sara Alex, Habibur Rahaman Khan, Subbaraya Gudde Ramachandra, Rudraiah Medhamurthy. Journal of the Endocrine Society (07 June 2023), DOI:10.1210/jendso/bvad076

Seed treatment with neonicotinoid insecticides does not affect the foraging behavior of honey bees” K. Chandrakumara, K. Muralimohan, Anand H. S., Suresh Gundoju, V. V. Belavadi & T. M. Ramanappa. Springer Link (15 May 2023), DOI:10.1007/s13592-023-01007-x

Role of intraluteal and intrauterine prostaglandin signaling in LH-induced luteolysis in pregnant rats” Akshi Vashistha, Habibur Rahaman Khan. Wiley Online Library (02 March 2023), DOI: 10.1002/mrd.23678

A New Antidiabetic Agent Showing Short- and Long-Term Effects Due to Peroxisome Proliferator-Activated Receptor Alpha/Gamma Dual Agonism and Mitochondrial Pyruvate Carrier Inhibition“, Antonio Laghezza, Carmen Cerchia, Massimo Genovese, Rosalba Leuci, Erica Pranzini, Alice Santi, Leonardo Brunetti, Luca Piemontese, Paolo Tortorella, Abanish Biswas, Ravi Pratap Singh, Suhas Tambe, Sudeep CA, Ashok Kumar Pattnaik, Venkatesan Jayaprakash, Paolo Paoli, Antonio Lavecchia, and Fulvio Loiodice. Journal of Medicinal Chemistry (2023), DOI:10.1021/acs.jmedchem.2c02093

Scientific and Regulatory Policy Committee Points to Consider for Medical Device Implant Site Evaluation in Nonclinical Studies” Maureen T. O’Brien, JoAnn C. L. Schuh, Lyn M. Wancket, Sarah D. Cramer, Kathleen A. Funk, Nicolette D. Jackson, Kamala Kannan, Kevin Keane, Abraham Nyska, Serge D. Rousselle, Adrienne Schucker, Valerie S. Thomas, Stefan Tunev. Sage Journals (2022), 50 (4), DOI:10.1177/019262332211032

Design and synthesis of novel spirocyclic carboxylic acids as potent and orally bioavailable DGAT1 inhibitors and their biological evaluation” Summon Koul, Suresh Kurhade, Sandeep Bhosale, Keshav Naik, Videsh Salunkhe, Sudhir Ravula, Prasad Punde, Ravikumar Velayutham, Atul Tiwari, Daniela Ahl, Srividya Malkapuram, Vamsi Mudagala, Amol Raje, Dhananjay Umrani, Suhas Tambe, Poonam Patil, Umesh Singh, Debnath Bhuniya, Narayanan Hariharan, Kasim Mookhtiar. Science Direct (2022), 62, DOI:10.1016/j.bmcl.2022.128632

Mycobactin Analogues with Excellent Pharmacokinetic Profile Demonstrate Potent Antitubercular Specific Activity and Exceptional Efflux Pump Inhibition“, Mousumi Shyam, Harshita Verma, Gourab Bhattacharje, Piyali Mukherjee, Samsher Singh, Sujit Kamilya, Pushpendu Jalani, Swetarka Das, Arunava Dasgupta, Abhishake Mondal, Amit Kumar Das, Amit Singh, Federico Brucoli, Claire Bagnéris, Rachael Dickman, Vinay N. Basavanakatti, Patibandla Naresh Babu, Vadivelan Sankaran, Abhimanyu Dev, Barij Nayan Sinha, Sanjib Bhakta, and Venkatesan Jayaprakash. Journal of Medicinal Chemistry (2022), 65(1), 234-256, DOI:10.1021/acs.jmedchem.1c01349

A sprayable Acid-Oxidizing solution containing hypochlorous acid (AOS2020) efficiently and safely inactivates SARS-Cov-2: a new potential solution for upper respiratory tract hygiene“, Nadia Giarratana, Balan Rajan, Kannan Kamala, Michelle Mendenhall & Giorgio Reiner. European Archives of Oto-Rhino-Laryngology (2021), DOI:10.1007/s00405-021-06644-5

Pharmacokinetics and Pharmacodynamic Herb-Drug Interaction of Piperine with Atorvastatin in Rats“, Thomas Asha B; Choudhary Durga C; Raje Amol; Nagrik Shatrughna S. Journal of Chromatographic Science (2021), 59 (4), DOI: 10.1093/chromsci/bmaa126

Scope of adjuvant therapy using roflumilast, a PDE-4 inhibitor against COVID-19“, Sugin Lal Jabaris S, Ranju V, DOI: 10.1016/j.pupt.2020.101978

A Series of Ferulic Acid Amides Reveals Unexpected Peroxiredoxin 1 Inhibitory Activity with in vivo Antidiabetic and Hypolipidemic Effects“, Yasmin Sabina; Cerchia Carmen; Badavath Vishnu Nayak; Lavecchia Antonio; Fabrizio Dal Piaz; Mondal K. Susanta; Atlı Özlem; Baysal Merve; Vadivelan Sankaran; Shankar S; Siddique Mohd Usman Mohd; Pattnaik Ashok Kumar; Singh Ravi Pratap; Loiodice Fulvio; Jayaprakash Venkatesan; Laghezza Antonio. ChemMedChem, 16 (3), DOI: doi.org/10.1002/cmdc.202000564

“Initial impurity screening for 5-batch analysis studies”, Vasireddi, Pardhasaradhi; Gogineni, Ravikant. Abstracts of Papers, 260th ACS National Meeting & Exposition, San Francisco, CA, United States, August 23-27, 2020 (2020), AGRO-0169

“Process for the preparation of Chlorantraniliprole”, Ashwin, V.; Pradhan, Ashok Kumar; Palimkar, Sanjay Sambhajirao; Mane, Avinash Sheshrao

In vitro drug metabolism and pharmacokinetics of a novel thiazolidinedione derivative, a potential anticancer compound“, Shankar, S.; Vuppu, Suneetha. Journal of Pharmaceutical and Biomedical Analysis (2020), 179, 113000. DOI:10.1016/j.jpba.2019.113000

A toxicogenomic approach for the risk assessment of the food contaminant acetamide“, Rance Nault, Bryan Bals, Farzaneh Teymouri, Michael B. Black, Melvin E. Andersen, Patrick D. McMullen, Seetha Krishnan, Nagesh Kuravadi, Neetha Paul, Santhosh Kumar, Kamala Kannan, K.C. Jayachandra, Lakshmanan Alagappan, Bhavesh Dhirajlal Patel, Kenneth T. Bogen, Bhaskar B. Gollapudi, James E. Klaunig, Tim R. Zacharewski, Venkataraman Bringi, Journal of Toxicology and Applied Pharmacology, Volume 388, Article ID 114872. DOI: 10.1016/j.taap.2019.114872

Capillary microsampling in mice: effective way to move from sparse sampling to serial sampling in pharmacokinetics profiling“, Raje, Amol A.; Mahajan, Vallabh; Pathade, Vishal V.; Joshi, Kaushal; Gavali, Ashutosh; Gaur, Ashwani; Kandikere, Vishwottam. Xenobiotica (2019), Ahead of Print. DOI:10.1080/00498254.2019.1683259

Response to comments on “Reproductive toxicology studies supporting the safety of molindone, a dopamine receptor antagonist”“, Gopalakrishnan Gopakumar; Ganiger Shivaputhrappa; White Tacey E K; Yu Chungping, Birth defects research (2019), 111(4), 230-231. DOI: 10.1002/bdr2.1447

b-Lactam based α-amino and α-hydroxy phosphonate ester molecular hybrids: synthesis, docking Studies and evaluation of anti-microbial activity against various gram-positive and gram-negative species“, Vangala, Vijaya Bhaskar; Pati, Hari N. International Journal of Pharmaceutical Sciences Review and Research (2019), 55(1), 34-40.

Development and validation of a chiral LC-ESI-MS/MS method for simultaneous determination of the enantiomeric metabolites isosorbide 2-mononitrate and isosorbide 5-mononitrate of isosorbide dinitrate in rat and human plasma“, Patel, Bhavesh D.; Pulakundam, Nageswararao; Gadekar, Ajit R.; Raje, Amol A.; Ramanathan, Vikram; Ameta, Rakshit. Journal of Pharmaceutical and Biomedical Analysis (2019), 174, 396-405. DOI:10.1016/j.jpba.2019.06.007

A simple and sensitive LC-MS/MS method for quantification of Bepridil in rat plasma and its application to pharmacokinetic studies“, Patel, Bhavesh D.; Palakundam, Nageswararao; Alamanda, Rajesh; Gadekar, Ajit R.; Raje, Amol A.; Ameta, Rakshit. Journal of Pharmaceutical and Biomedical Analysis (2019), 172, 113-119. DOI:10.1016/j.jpba.2019.04.038

Discovery and evaluation of novel FAAH inhibitors in neuropathic pain model“, Bhuniya, Debnath; Kharul, Rajendra K.; Hajare, Atul; Shaikh, Nadim; Bhosale, Sandeep; Balwe, Sandip; Begum, Fouzia; De, Siddhartha; Athavankar, Sonalee; Joshi, Dhananjay; et al. Bioorganic & Medicinal Chemistry Letters (2019), 29(2), 238-243. DOI:10.1016/j.bmcl.2018.11.048

Recombinant irisin induces weight loss in high fat DIO mice through increase in energy consumption and thermogenesis“, Niranjan Sanjay B; Belwalkar Shraddha Vijay; Tambe Suhas; Venkataraman Krishnan; Mookhtiar Kasim A. Biochemical and biophysical research communications (2019), 519(2), 422-429. DOI:10.1016/j.bbrc.2019.08.112

Herb-Drug Interaction of Quercetin on the Pharmacokinetics of Losartan in Rats: A High-Performance Thin-Layer Chromatography Study“, Shraddha Jadhao, Asha Thomas, Amol Raje, Shatrughna Nagrik, Lata Kothapalli, Aaftab Shaikh. JPC – Journal of Planar Chromatography – Modern TLC (2019), 32(5), 401–409. DOI:10.1556/1006.2019.32.5.8

Development and validation of LC-MS/MS method for determination of DNDI-VL-2098 in mouse, rat, dog and hamster blood“, Patel Bhavesh D; Uppal Ritika; Pulakundam Nageswararao; Patel Jignesh P; Ramanathan Vikram;. Bioanalysis (2019), 11(15), 1419-1435. DOI:10.4155/bio-2019-0128

The food contaminant acetamide is not an in vivo clastogen, aneugen, or mutagen in rodent hematopoietic tissue“, Moore Martha M; Gollapudi Bhaskar; Nagane Rajendra; Khan Nadeem; Patel Manish; Khanvilkar Tushar; Roy Avani M; Ramesh E; Bals Bryan; Teymouri Farzaneh; et al. Regulatory toxicology and pharmacology : RTP (2019), 108104451. DOI:10.1016/j.yrtph.2019.104451

Discovery and pharmacological evaluation of indole derivatives as potent and selective RORγt inverse agonist for multiple autoimmune conditions“, Shaikh Nadim S; Iyer Jitesh P; Munot Yogesh S; Mukhopadhyay Partha P; Raje Amol A; Nagaraj Ranganayaki; Jamdar Vijay; Gavhane Ravindra; Lohote Mahendra; Sherkar Prasad; et al. Bioorganic & medicinal chemistry letters (2019), 29(16), 2208-2217. DOI:10.1016/j.bmcl.2019.06.044

Validation of a sensitive simultaneous LC-MS/MS method for the quantification of novel anti-cancer thiazolidinedione and quinazolin-4-one derivatives in rat plasma and its application in a rat pharmacokinetic study“, Shankar Sengottuvelan, Ritika Uppala, Suneetha Vuppub, Journal of Chromatography B, Volume 1121, 15 July 2019, Pages 18-27; DOI: 10.1016/j.jchromb.2019.05.003

Lyophilized B. subtilis ZB183 Spores: 90-Day Repeat Dose Oral (Gavage) Toxicity Study in Wistar Rats“, B. Appala Naidu, Kamala Kannan, D. P. Santhosh Kumar, John W. K. Oliver and Zachary D. Abbott, Hindawi, Journal of Toxicology, Volume 2019, Article ID 3042108, 9 pages; DOI: 10.1155/2019/3042108

Sustainable Amine Synthesis: Iron Catalyzed Reactions of Hydrosilanes with Imines, Amides, Nitroarenes and Nitriles“, Nadim S. Shaikh, Chemistry Select, 4(22), 6753-6777, DOI: 10.1002/slct.201900460

Luminescent bis(benzo[d]thiazolyl)quinoxaline: facile synthesis, nucleic acid and protein BSA interaction, live-cell imaging, biopharmaceutical research and cancer theranostic application†“, Lavanya Thilak Babu, Gajanan Raosaheb Jadhav and Priyankar Paira, RSC Advance, 2019,9, 8748-8752, DOI: 10.1039/C9RA01498E

Cytotoxic 2‐(2′‐Hydroxyphenyl)benzothiazolylquinoline Analogues and their In Vitro Screening through Developmental Assays†“, Gajanan Raosaheb Jadhav, Dr. Priyankar Paira, Chemistry Select, 4(12), 3524-3530, DOI: 10.1002/slct.201803618

Reproductive Toxicology Studies Supporting the Safety of Molindone, a Dopamine Receptor Antagonist“, Gopalakrishnan G, Ganiger S, White TEK, Yu C. Reproductive toxicology studies supporting the safety of molindone, a dopamine receptor antagonist. Birth Defects Research.2018; e1381, DOI: 10.1002/bdr2.1381

Acute Histopathologic Findings Related to Needle Puncture Trauma during Subcutaneous Injection in the Sprague-Dawley Rat Model“,Ramot Yuval; Kannan Kamala; Reddy Sathish; Krishnappa H; Dillberger John E; Nyska Abraham. Toxicologic pathology (2018), 47(1), 93-96. DOI:10.1177%2F0192623318808989

In-vitro metabolism, CYP profiling and metabolite identification of E- and Z- guggulsterone, a potent hypolipidmic agent“, Chhonker Yashpal S; Chandasana Hardik; Bala Veenu; Mukkavilli Rao; Kumar Deepak; Vangala Subrahmanyam; Bhatta Rabi S. Journal of pharmaceutical and biomedical analysis (2018), 160202-211. DOI:10.1016/j.jpba.2018.06.047

Toxicity and toxicokinetic study of RPh201 in Sprague-Dawley rats“, Ramot Yuval; Hazan Zadik; Lucassen Andre; Adamsky Konstantin; Santhosh Kumar D P; Vijayasarathi S K; Krishnappa H; Seervi Madhav Singh; Nyska Abraham. Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association (2018), 112168-177. DOI:10.1016/j.fct.2017.12.036

Efficient synthesis of β-lactam-containing α-aminophosphonates using fumaric acid as mild catalyst, Vangala, Vijaya Bhaskar; Pati, Hari Narayan
Chemical Methodologies (2018), 2(4), 333-340. DOI:10.22034/chemm.2018.66128

Isoxazole-Tethered Diarylheptanoid Analogs: Discovery of a New Drug-like PAR2 Antagonist“, Bhuniya, Debnath; Bhosale, Sandeep; Reddy, Satyanarayana B.; Reddy, Sudharshan N., Bioorganic & Medicinal Chemistry Letters (2018), 28(13), 2285-2288, DOI: 10.1016/j.bmcl.2018.05.032

Safety evaluation of fructooligosaccharide (FOSSENCETM): Acute, 14-day, and subchronic oral toxicity study in Wistar rats”, Manish Jain, Manoj Gote, Ashok Kumar Dubey, S Narayanan, H. Krishnappa, DP Santhosh Kumar, GS Ravi, SK Vijayasarathi, and S Shankar, J. Toxicology Research and Application, 2018, 2, DOI: 10.1177/2397847318787750

The Pathology Community’s Interpretation of Settiagounder’s Proposals on GLP Process as Applied to Pathology Peer Review”, Natesan Settiagounder. Letter to the Editor. J. Regulatory Science, 2018, 6 (1), xii – xix

Histopathology peer review process. The compliance conundum“. Natesan Settiagounder, Quasar, 2018, 143, 20 – 25

Assessing Drug Interaction Potential of Herbal Medicine Liv.52, Smokeless Tobacco Snuff and Edible Camphor using Human Liver Microsomes“. Rao Mukkavilli, Gajanan Jadhav, Shankar Sengottuvelan and Subrahmanyam Vangala, EC Pharmacology and Toxicology, 6(4) (2018): 277-290

Evaluation of separate role of intestine and liver in first pass metabolism of budesonide in rat“. Amol A Raje, Radni D Deshpande, Vishal V Pathade, Vallabh Mahajan, Kaushal Joshi, Ashwini Tambe, Ramana Jinugu, Vamsi L M Madgula, Ashwani Gaur, Vishwottam Kandikere, Chandragouda R Patil, Kasim A Mookhtiar, Xenobiotica, 48(12):1206-1214. DOI: 10.1080/00498254.2017.1404168.

Evaluation of Drug Transport in MDCKIIWild Type, MDCKIIMDR1, MDCKIIBCRP and Caco2 Cell Lines Mukkavilli“, Mukkavilli, Rao; Jadhav, Gajanan; Vangala, Subrahmanyam. J. Pharmaceutical Biotechnology (2017), 18(14), 1151-1158. DOI: 10.2174/1389201019666180308091855

Discovery and evaluation of 1H-pyrrolo[2,3-b]pyridine based selective and reversible small molecule BTK inhibitors for the treatment of rheumatoid arthritis.“, Thakkar, Mahesh; Bhuniya, Debnath; Kaduskar, Rahul; Mengawade, Tanaji; Naik, Keshav; Salunkhe, Videsh; Bhalerao, Amit; Kurhade, Santosh; Mavinahalli, Jagadeesh; Jain, Vaibhav. By et al From Bioorganic & Medicinal Chemistry Letters (2017), 27(8), 1867-1873. DOI: 10.1016/j.bmcl.2017.02.026

Basics of Stem Cells and Preclinical Testing“, K. Suryanarayana Rao, Biology, Engineering, Medicine and Science Reports, 2017,3,1,13-16, DOI : 10.5530/bems.3.1.5

Practical Considerations in the Conduct of Micronucleus Test“, K. Suryanarayana Rao, Biology, Engineering, Medicine and Science Reports, 2017,3,1,11-12, DOI : 10.5530/bems.3.1.4

Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson’s Disease and Depression”, Sujay Basu; Dinesh A. Barawkar; Vidya Ramdas; Minakshi Naykodi; Yogesh D. Shejul; Meena Patel; Sachin Thorat; Anil Panmand; K. Kashinath; Rajesh Bonagiri; Vandna Prasad; Ganesh Bhat; Azfar Quraishi; Sumit Chaudhary; Amol Magdum; Ashwinkumar V. Meru; Indraneel Ghosh; Ravi K. Bhamidipati; Amol A. Raje; Vamsi L. M. Madgula; Siddhartha De; Sreekanth R. Rouduri; Venkata P. Palle; Anita Chugh; Narayanan Hariharan; Kasim A. Mookhtiar, ACS Medicinal Chemistry Letters, 2017, 8, 835−840, DOI: 10.1021/acsmedchemlett.7b00175

Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation”, Basu, Sujay; Barawkar, Dinesh A.; Thorat, Sachin; Shejul, Yogesh D.; Patel, Meena; Naykodi, Minakshi; Jain, Vaibhav; Salve, Yogesh; Prasad, Vandna; Chaudhary, Sumit; Ghosh, Indraneel; Bhat, Ganesh; Quraishi, Azfar; Patil, Harish; Ansari, Shariq; Menon, Suraj; Unadkat, Vishal; Thakare, Rhishikesh; Seervi, Madhav S.; Meru, Ashwinkumar V.; De, Siddhartha; Bhamidipati, Ravi K.; Rouduri, Sreekanth R.; Palle, Venkata P.; Chug, Anita; Mookhtiar, Kasim, Journal of Medicinal Chemistry , 60, 2,681-694

Safety evaluation of galactooligosaccharides: Subchronic oral toxicity study in Sprague-Dawley rats”, Toxicology Research and Application ,1, 1-12

Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases”, Sujay Basu, Dinesh A. Barawkar, Vidya Ramdas, Meena Patel, Yogesh Waman, Anil Panmand, Santosh Kumar, Sachin Thorat, Minakshi Naykodi, Arnab Goswami, B. Srinivasa Reddy, Vandna Prasad, Sandhya Chaturvedi, Azfar Quraishi, Suraj Menon, Shalini Paliwal, Abhay Kulkarni, Vikas Karande, Indraneel Ghosh, Syed Mustafa, Siddhartha De, Vaibhav Jain, Ena Ray Banerjee, Sreekanth R. Rouduri, Venkata P. Palle, Anita Chugh, Kasim A. Mookhtiar, European journal of medicinal chemistry ,134 ,218-229

Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors”, Basu, Sujay; Prathipati, Philip; Thorat, Sachin; Ansari, Shariq; Patel, Meena; Jain, Vaibhav; Jinugu, Ramana R.; Niranjan, Sanjay; De, Siddhartha; Reddy, Satyanarayana, Bioorganic & Medicinal Chemistry, 25, 1, 67-74

A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives”, Basu, Sujay; Barawkar, Dinesh A.; Ramdas, Vidya; Waman, Yogesh; Patel, Meena; Panmand, Anil; Kumar, Santosh; Thorat, Sachin; Bonagiri, Rajesh; Jadhav, Dilip; Mukhopadhyay, Partha; Prasad, Vandna; Reddy, B. Srinivasa; Goswami, Arnab; Chaturvedi, Sandhya; Menon, Suraj; Quraishi, Azfar; Ghosh, Indraneel; Dusange, Sushant; Paliwal, Shalini; Kulkarni, Abhay; Karande, Vikas; Thakre, Rhishikesh; Bedse, Gaurav; Rouduri, Sreekanth; Gundu, Jayasagar; Palle, Venkata P.; Chugh, Anita; Mookhtiar, Kasim A., European journal of medicinal chemistry , 127, 986-996

Histopathology Evaluation and Peer Review for Nonclinical Studies: Raw Data Compliance to GLP Quality Systems“, Settiagounder, Natesan, Journal of Regulatory Science, 2017, 5, 2, 45-55

Histopathology Peer Review for Nonclinical Studies – GLP Processes and Conditions“, Settiagounder, Natesan, Journal of Regulatory Science, 2017, 5, 2, 56-66

In vitro and in vivo anticancer activity of 2-acetyl-benzylamine isolated from Adhatoda vasica L. leaves“, C. Balachandran, Y. Arun, B. Sangeethac, V. Duraipandiyan, S. Awale, N. Emi, S. Ignacimuthu, P. T. Perumal, Biomedicine & Pharmacotherapy, 2017, 93, 96-806, DOI:10.1016/j.biopha.2017.06.096.

Modifications of flexible nonyl chain and nucleobase head group of (+)-erythro-9-(2′s-hydroxy-3′s-nonyl)adenine [(+)-EHNA] as adenosine deaminase inhibitors“, Sachin R.Kandalkar, Parimi Atchuta Ramaiah, Manoj Joshi, Atul Wavhal, Yogesh Waman, Amol A.Raje, Ashwini Tambe, Shariq Ansari, Siddhartha De, Venkata P.Palle, Kasim A.Mookhtiar, Anil M.Deshpande, Dinesh A.Barawkara, Bioorganic & Medicinal Chemistry, 2017, 25(2), 5799-5819, DOI:10.1016/j.bmc.2017.09.015.

Discovery of liver-directed glucokinase activator having anti-hyperglycemic effect without hypoglycemia“, Anil M. Deshpande, Debnath Bhuniya, Siddhartha De, Bhavesh Dave, Vinod P. Vyavahare, Santosh H. Kurhade, Sachin R. Kandalkar, Keshav P. Naik, Balasaheb S.Kobal, Rahul D. Kaduskar, Sujay Basu, Vaibhav Jain, Pratima Patil, Sandhya Chaturvedi Joshi, Ganesh Bhat, Amol A. Raje, Satyanarayana Reddy, Jayasagar Gundu, Vamsi Madgula, Suhas Tambe, Prasad Shitole, Dhananjay Umrani, Anita Chugh, Venkata P.Palle, Kasim A. Mookhtiar, European Journal of Medicinal Chemistry, 2017, 133, 268-286, DOI:10.1016/j.ejmech.2017.03.042.

Design and synthesis of novel, potent and selective hypoxanthine analogs as adenosine A 1 receptor antagonists and their biological evaluation“, Summon Koul, Vidya Ramdas, Dinesh A Barawkar, Yogesh B Waman, Neela Prasad, Santosh Kumar Madadi, Yogesh D Shejul, Rajesh Bonagiri, Sujay Basu, Suraj Menon, Srinivasa B Reddy, Sandhya Chaturvedi, Srinivas Rao Chennamaneni, Gaurav Bedse, Rhishikesh Thakare, Jayasagar Gundu, Sumit Chaudhary, Siddhartha De, Ashwinkumar V Meru, Venkata Palle, Anita Chugh, Kasim A Mookhtiar, Bioorg Med Chem., 2017, 25(6), 1963-1975, DOI:10.1016/j.bmc.2017.02.029.

Development of a Scalable Process for the Synthesis of DNDI-VL-2098: A Potential Preclinical Drug Candidate for the Treatment of Visceral Leishmaniasis“, Vijay S. Satam, Srinivasa Rao Pedada, Pasumpon Kamaraj, Nakita Antao, Apoorva Singh, Rama Mohan Hindupur, Hari N. Pati, Andrew M. Thompson, Delphine Launay, Denis Martin, Organic Process Research & Development, 2017, 21(1), 52–59, DOI:10.1021/acs.oprd.6b00331.

“Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors”, Basu, Sujay; Prathipati, Philip; Thorat, Sachin; Ansari, Shariq; Patel, Meena; Jain, Vaibhav; Jinugu, Ramana R.; Niranjan, Sanjay; De, Siddhartha; Reddy, Satyanarayana, Bioorganic & Medicinal Chemistry, 2016, DOI: 10.1016/j.bmc.2016.10.012

“Identification, charecterization and quantification of process related impurities in azimsulfuron technical”, Venkatesh, M. Prabhu; Pardhasaradhi, V.; Dhayanithi, V.; Avinash, Mane; Palimkar, S.; Subhash, R. Kadam; Mohan, Hindupur Rama, Chemical Science Transactions, 2016, 5, 1, 41-55, DOI: 10.7598/cst2016.1132

“Impact of APCI ionization source in liquid chromatography tandem mass spectrometry based tissue distribution studies”, Khatal Laxman; Gaur Ashwani; Naphade Ashish; Kandikere Vishwottam; Mookhtiar Kasim, Biomedical chromatography : BMC, 2016, 30, 10, 1676-85

“Isolation and characterization of 2-hydroxy-9,10-anthraquinone from Streptomyces olivochromogenes (ERINLG-261) with antimicrobial and antiproliferative properties”, Chandrasekar Balachandran, Veeramuthu Duraipandiyan, Yuvaraj Arun, Balachandran Sangeetha, Nobuhiko Emi, Naif Abdullah Al-Dhabi, Savarimuthu Ignacimuthu, Yoko Inaguma Akinao Okamoto, Paramasivan T.Perumal. Revista Brasileira de Farmacognosia (2016), 26(3), 285-295. DOI: 10.1016/j.bjp.2015.12.003

“Assessment of in vitro metabolic stability, plasma protein binding, and pharmacokinetics of E- and Z-guggulsterone in rat”, Chhonker Yashpal S; Chandasana Hardik; Prasad Yarra Durga; Laxman Tulsankar Sachin; Bhatta Rabi S; Chhonker Yashpal S; Chandasana Hardik; Laxman Tulsankar Sachin; Bhatta Rabi S; Mukkavilli Rao; Vangala Subrahmanyam; Mukkavilli Rao, Drug testing and analysis, 2016, 8, 9, 966-75

“Effects of Gymnema sylvestre extract on the pharmacokinetics and pharmacodynamics of glimepiride in streptozotocin induced diabetic rats”, Kamble Bhagyashree;  Gupta Ankur; Moothedath Ismail; Duraiswamy B;  Khatal Laxman; Janrao Shirish; Jadhav Amol, Chemico-biological interactions, 2016,  24530-8

“Efficient synthesis of β-lactam containing α-hydroxy phosphonates using tartaric acid and fumaric acid as mild catalysts”, Vangala, Vijaya Bhaskar; Pati, Hari N., Synthetic Communications 2016, 46, 4, 374-378, DOI:10.1080/00397911.2016.1139722

“Synthesis and antiproliferative properties of isoxazole analogs containing dibenzosuberane moiety”,  Moger, Manjunath; Pradhan, Ashok; Singh, Apoorva; Govindaraju, Darshan Raj Chenna; Hindupur, Rama Mohan; Pati, Hari N., Medicinal Chemistry Research 2016, 25, 3, 449-455, DOI:10.1007/s00044-015-1497-3

“Protective role of liv.52 on the toxicity of acetaminophen during embryogenesis in Wistar rats”, Santhosh Kumar, D.P., Deecaraman, M., Vijayalaksmi, M., Ramesh Edamula, Krishnappa, H., Latha, M. and GeethaRao, G, International Journal of Current Research, 2015, 7, 5, 16392-16401, ISSN:0975-833X

“Pharmacological and Biological Activities of Benzazepines: An Overview”, Shah, Jigar H.; Hindupur, Rama M.; Pati, Hari N., Current Bioactive Compounds, 2015, 11, 3, 170-188, DOI:10.2174/1573407211666150910202200

“Aminothiazoles: Hit to lead development to identify antileishmanial agents”, Bhuniya, Debnath; Mukkavilli, Rao; Shivahare, Rahul; Launay, Delphine; Dere, Ravindra T.; Deshpande, Anil; Verma, Aditya; Vishwakarma, Preeti; Moger, Manjunath; Pradhan, Ashok; et al, European Journal of Medicinal Chemistry (2015), 102, 582-593, DOI:10.1016/j.ejmech.2015.08.013

“Efficient and Scalable Process for Synthesis of 5-Nitro-7-azaindole”, Bhat, Prasanna V.; Dere, Ravindra T.; Ravikumar, S.; Hindupur, Rama Mohan; Pati, Hari N., Organic Process Research & Development, 2015, 19, 9, 1282-1285., DOI:10.1021/acs.oprd.5b00181

“Preparation of substituted heterobicyclic compounds, compositions and medicinal applications thereof”, Thakkar, Mahesh; Koul, Summon; Bhuniya, Debnath; Mookhtiar, Kasim, Indian Pat. Appl., 2015, IN 2012CH01573 A 20150710

“Chemistry of macrocyclic β-lactam: an overveiw”, Vangala, Vijaya Bhaskar; Maddani, Mahagundappa Rachappa; Hindupur, Rama Mohan; Pati, Hari Narayan,  Heterocycles, 2015, 91, 4, 701-717, DOI:10.3987/REV-14-812

“Noscapine recirculates enterohepatically and induces self-clearance”, Mukkavilli, Rao; Gundala, Sushma R.; Yang, Chunhua; Jadhav, Gajanan R.; Vangala, Subrahmanyam; Reid, Michelle D.; Aneja, Ritu, European Journal of Pharmaceutical Sciences, 2015, 77, 90-99, DOI:10.1016/j.ejps.2015.05.026

“Identification and Synthesis of Major Impurities Formed During the Synthesis of Trifloxystrobin and Kresoxim- methyl Fungicides”, Kamaraj, Pasumpon; Antao, Nakita; Singh, Apoorva; Satam, Vijay; Kadam, Subhash; Prabhu, Venkatesh M.; Hindupur, Rama Mohan; Pati, Hari N., Letters in Organic Chemistry, 2015, 12, 5, 306-310, DOI:10.2174/1570178612666150318002831

“Preparation of substituted heterobicyclic compounds, compositions and medicinal applications thereof as Btk inhibitors”,  Thakkar, Mahesh; Koul, Summon; Bhuniya, Debnath; Mookhtiar, Kasim; Kurhade, Santosh; Munot, Yogesh; Mengawade, Tanaji; Kulkarni, Bheemashankar A., From U.S. Pat. Appl. Publ., 2015, US 20150064196 A1 20150305

“A process for the preparation of fluoxastrobin”, Hindupur, Rama Mohan; Mane, Avinash Sheshrao; Balakrishnan, Sankar; Pawar, Jivan Dhanraj; Maddani, Mahagundappa Rachappa; Wadhwa, Sandeep; Prasad, Vic, U.S. Pat. Appl. Publ., 2015, US 20150011753 A1 20150108

“Assessment of in vitro metabolic stability, plasma protein binding, and pharmacokinetics of E- and Z- guggulsterone in rat”, Chhonker Yashpal S; Chandasana Hardik; Prasad Yarra Durga; Laxman Tulsankar Sachin; Bhatta Rabi S; Chhonker Yashpal S; Chandasana Hardik; Laxman Tulsankar Sachin; Bhatta Rabi S; Mukkavilli Rao; et al, Drug testing and analysis, 2015

“In vitro anticancer activity of methyl caffeate isolated from Solanum torvum Swartz. Fruit”, Balachandran C; Emi N; Yamamoto Y; Inaguma Yoko; Okamoto Akinao; Arun Y; Perumal P T; Ahilan B; Ignacimuthu S; Sangeetha B; et al, Chemico-biological interactions, 2015, 24281-90

“Reversibility of dopamine receptor antagonist-induced hyperprolactinemia and associated histological changes in Tg RasH2 wild-type mice”, Krishna Gopala; Gopalakrishnan Gopa; Goel Saryu; Ganiger Shivaputhrappa; Kannan Kamala, Reproductive toxicology, 2015, 5873-8

“Noscapine recirculates enterohepatically and induces self-clearance”, Mukkavilli Rao; Gundala Sushma R; Yang Chunhua; Jadhav Gajanan R; Vangala Subrahmanyam; Reid Michelle D; Aneja Ritu, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences , 2015, 7790-9

“Synergistic interactions among flavonoids and acetogenins in Graviola (Annona muricata) leaves confer protection against prostate cancer”, Yang Chunhua; Gundala Sushma Reddy; Aneja Ritu; Mukkavilli Rao; Vangala Subrahmanyam; Reid Michelle D., Carcinogenesis, 2015, 36, 6, 656-65

“A convenient and mild one pot synthesis of cyclopentenone derivatives”, Moger, Manjunath; Pradhan, Ashok Kumar; Hindupur, Rama Mohan; Pati, Hari N., Tetrahedron Letters,  2014, 55, 16, 2675-2678, DOI:10.1016/j.tetlet.2014.03.038

“A flavonoid isolated from Streptomyces sp. (ERINLG-4) induces apoptosis in human lung cancer A549 cells through p53 and cytochrome c release caspase dependant pathway”, Balachandran C; Ignacimuthu S; Balakrishna K; Sangeetha B; Duraipandiyan V; Raj M Karunai; Parthasarathy K; Al-Dhabi N A; Arasu M Valan; Arulmozhi N M, Chemico-biological interactions, 2014, 22424-35

“An efficient synthesis of new β-lactam substituted 1,2,3-triazole via CuI-NBS mediated Click Chemistry”, Vangala, Vijaya Bhaskar; Mane, Avinash S.; Hindupur, Rama Mohan; Pati, Hari N., Chemistry Journal 2014, 4, 1, 8-12, 5

“Cholesterol homeostasis: lipoproteins in action”, Malashetty, Vijaykumar B., Asian Journal of Science and Technology, 2014, 5, 7, 400-404

“Design, synthesis, ADME characterization and antileishmanial evaluation of novel substituted quinoline analogs”, Gopinath, Vadiraj S.; Rao, Mukkavilli; Shivahare, Rahul; Vishwakarma, Preeti; Ghose, Sweta; Pradhan, Ashok; Hindupur, Ramamohan; Sarma, Koushik Das; Gupta, Suman; Puri, Sunil K.; et al, Bioorganic & Medicinal Chemistry Letters, 2014, 24, 9, 2046-2052, DOI:10.1016/j.bmcl.2014.03.065

“Development and validation of a liquid chromatographic enantiomer separation method for the estimation of (S)-enantiomer in sitagliptin”, Mone, Mahesh Kumar; Jain, Payal; Kurhade, Santosh; Sonune, Dnyaneshwar P.; Kaduskar, Rahul D., International Journal of Pharmaceutical Sciences and Research, 2014, 5, 6, 2382-2386, DOI:10.13040/IJPSR.0975-8232.5(6).2382-86

“Enterohepatic recirculation of bioactive ginger phytochemicals is associated with enhanced tumor growth-inhibitory activity of ginger extract”, Gundala Sushma R; Yang Chunhua; Aneja Ritu; Mukkavilli Rao; Vangala Subrahmanyam; Yadav Pooja; Tandon Vibha; Prakash Satya, Carcinogenesis, 2014, 35, 6, 1320-9

“Hydroxychavicol, a betel leaf component, inhibits prostate cancer through ROS-driven DNA damage and apoptosis”, Gundala Sushma Reddy; Yang Chunhua; Paranjpe Rutugandha; Brahmbhatt Meera; Pannu Vaishali; Cheng Alice; Mukkavilli Rao; Reid Michelle D; Aneja Ritu, Toxicology and applied pharmacology, 2014, 280, 1, 86-96

“In vitro metabolism, disposition, preclinical pharmacokinetics and prediction of human pharmacokinetics of DNDI-VL-2098, a potential oral treatment for Visceral Leishmaniasis”, Mukkavilli, Rao; Pinjari, Jakir; Patel, Bhavesh; Sengottuvelan, Shankar; Mondal, Subodh; Gadekar, Ajit; Verma, Manas; Patel, Jignesh; Pothuri, Lavanya; Chandrashekar, Gopu; et al, European Journal of Pharmaceutical Sciences, 2014, 65, 147-155, DOI:10.1016/j.ejps.2014.09.006

“Cytomegalovirus pp65 limits dissemination but is dispensable for persistence”, Daniel Malouli, Scott G. Hansen, Ernesto S. Nakayasu, Emily E. Marshall, Colette M. Hughes, Abigail B. Ventura, Roxanne M. Gilbride, Matthew S. Lewis, Guangwu Xu, Craig Kreklywich, Nathan Whizin, Miranda Fischer, Alfred W. Legasse, Kasinath Viswanathan, Don Siess, David G. Camp II, Michael K. Axthelm, Christoph Kahl, Victor R. DeFilippis, Richard D. Smith, Daniel N. Streblow,1 Louis J. Picker, Klaus Früh1. JCI The Journal of Clinical Investigation, 2014, 124(5), 1928–1944, DOI: 10.1172/JCI67420.

“Modulation of cytochrome P450 metabolism and transport across intestinal epithelial barrier by ginger biophenolics”, Mukkavilli, Rao; Gundala, Sushma R.; Yang, Chunhua; Donthamsetty, Shashikiran; Cantuaria, Guilherme; Jadhav, Gajanan R.; Vangala, Subrahmanyam; Reid, Michelle D.; Aneja, Ritu, PLoS One, 2014, 9, 9, DOI:10.1371/journal.pone.0108386

“Novel third-generation water-soluble noscapine analogs as superior microtubule-interfering agents with enhanced antiproliferative activity”, Henary Maged; Owens Eric A; Nagaraju Mulpuri; Hamelberg Donald; Narayana Lakshminarayana; Yadav Yogesh; Ahad Shazia; Panda Dulal; Gundala Sushma R; Sharma Vibhuti; et al, Biochemical pharmacology, 2014, 92, 2, 192-205

“Preparation of spirocyclic compounds as DGAT1 inhibitors, compositions containing same, and medicinal applications thereof”, Koul, Summon; Bhuniya, Debnath; Mookhtiar, Kasim; Bhosale, Sandeep; Kurhade, Suresh; Naik, Keshav; Velayutham, Ravikumar; Salunkhe, Videsh, PCT Int. Appl., 2014, WO 2014054053 A1 20140410

“Preparation of substituted fused tricyclic compounds as JAK kinase inhibitors, compositions and medicinal applications thereof”, Barawkar, Dinesh; Bende, Tanushree; Zahler, Robert; Bandyopadhyay, Anish, Indian Pat. Appl., 2014, IN 2011CH00891 A 20140214

“Preparation of tricyclic compounds as JAK modulators for treatment of JAK-associated diseases”, Barawkar, Dinesh; Bandyopadhyay, Anish; Zahler, Robert; Sarangthem, Robindro; Waman, Yogesh; Bonagiri, Rajesh; Jadhav, Dilip; Mukhopadhyay, Partha, PCT Int. Appl., 2014, WO 2014045305 A1 20140327

“Synthesis and antimicrobial evaluation of some substituted-3-aryl-2,3,4,5,6,7-hexahydro-1H-inden-1-one”, Moger, Manjunath; Govndraju, Darshan Raj C.; Hindupur, Rama Mohan; Pati, Hari Narayan, Chemical Science Transactions, 2014, 3, 4, 1483-1487, 5 pp.,  DOI:10.7598/cst2014.867

“Synthesis and antimicrobial properties of 1,3,4-oxadiazole analogs containing dibenzosuberane moiety”, Moger, Manjunath; Satam, Vijay; Govindaraju, Darshan Raj C.; Paniraj, A. S.; Gopinath, Vadiraj S.; Hindupur, Rama Mohan; Pati, Hari N., Journal of the Brazilian Chemical Society, 2014, 25, 1, 104-111, DOI:10.5935/0103-5053.20130275

“Synthesis of L-azaisotryptophan and its analogs: a general access to new 2-substituted azaindoles”, Kurhade, Santosh; Rajopadhyay, Vandana; Avaragolla, Satheesh Veerappa; Koul, Summon; Ramaiah, Parimi Atchuta; Bhuniya, Debnath, Tetrahedron Letters, 2014, 55, 15, 2415-2419, DOI:10.1016/j.tetlet.2014.02.125

“Synthesis of substituted esters of imidazoles, oxazoles, thiazoles, and diethyl pyrazine-2,5-dicarboxylate from a common acyclic precursor employing C-formylation strategy”, Khose, Goraksha; Shinde, Shailesh; Panmand, Anil; Kulkarni, Ravibhushan; Munot, Yogesh; Bandyopadhyay, Anish; Barawkar, Dinesh; Patil, Santoshkumar N., Tetrahedron Letters, 2014, 55, 16, 2671-2674, DOI:10.1016/j.tetlet.2014.03.039

“An Improved Kilogram-Scale Synthesis of 2-Bromo-4-nitro-1H-imidazole: A Key Building Block of Nitroimidazole Drugs”, Pedada, Srinivasa Rao; Satam, Vijay S.; Tambade, Pawan J.; Kandadai, Srinivas A.; Hindupur, Rama Mohan; Pati, Hari N.; Launay, Delphine; Martin, Denis, Organic Process Research & Development, 2013, 17, 9, 1149-1155, DOI:10.1021/op400095f

“Design, synthesis and biological evaluation of 2-substituted quinolines as potential antileishmanial agents”, Gopinath, Vadiraj S.; Pinjari, Jakir; Dere, Ravindra T.; Verma, Aditya; Vishwakarma, Preeti; Shivahare, Rahul; Moger, Manjunath; Kumar Goud, Palusa Sanath; Ramanathan, Vikram; Bose, Prosenjit; et al, European Journal of Medicinal Chemistry, 2013, 69, 527-536, DOI:10.1016/j.ejmech.2013.08.028

“Highly efficient one-pot amination of carboxylate-substituted nitrogen-containing heteroaryl chlorides via Staudinger reaction”, Kandalkar, Sachin R.; Kaduskar, Rahul D.; Ramaiah, Parimi Atchuta; Barawkar, Dinesh A.; Bhuniya, Debnath; Deshpande, Anil M., Tetrahedron Letters, 2013, 54, 5, 414-418., DOI:10.1016/j.tetlet.2012.11.027

“Isolation, characterization of degradation products of sitagliptin and development of validated stability-indicating HPLC assay method for sitagliptin API and tablets”,  Sonune, Dnyaneshwar P.; Mone, Mahesh Kumar, International Journal of Pharmaceutical Sciences and Research, 2013, 4, 9, 3494-3503, 10,  DOI:10.13040/IJPSR.0975-8232.4(9).3494-03

“Preparation of amide compounds as FAAH inhibitors, compositions and applications thereof”, Kharul, Rajemdra; Bhuniya, Debnath; Mookhtiar, Kasim; Singh, Umesh; Hazare, Atul; Patil, Satish; Datrange, Laxmikant; Thakkar, Mahesh, Indian Pat. Appl., 2013, IN 2011CH03308 A 20130621

“Preparation of amide compounds as FAAH inhibitors, compositions and applications thereof”, Kharul, Rajendra; Bhuniya, Debnath; Mookhtiar, Kasim A.; Singh, Umesh; Hazare, Atul; Patil, Satish; Datrange, Laxmikant; Thakkar, Mahesh, PCT Int. Appl., 2013, WO 2013042139 A1 20130328

“Preparation of fused tricyclic compounds as therapeutic adenosine receptor antagonists”, Barawkar, Dinesh; Basu, Sujay; Ramdas, Vidya, Indian Pat. Appl., 2013, IN 2010CH02808 A 20130329

“Preparation of substituted heterobicyclic compounds, compositions and medicinal applications thereof”, Thakkar, Mahesh; Koul, Summon; Bhuniya, Debnath; Singh, Umesh, PCT Int. Appl., 2013, WO 2013157021 A1 20131024

“Preparation of substituted heterobicyclic compounds, compositions and medicinal applications thereof”, Thakkar, Mahesh; Koul, Summon; Bhuniya, Debnath; Mookhtiar, Kasim; Kurhade, Santosh; Munot, Yogesh, PCT Int. Appl., 2013, WO 2013157022 A1 20131024

“Stereo-controlled total syntheses of ieodomycins A and B using D-glucose based chiral pool approach”, Salunkhe, Videsh T.; Bhosale, Sandeep; Punde, Prasad; Bhuniya, Debnath; Koul, Summon, Tetrahedron Letters, 2013, 54, 20, 2489-2491, DOI:10.1016/j.tetlet.2013.03.002

“Synthesis of a sex pheromone of the longtailed mealybug, Pseudococcus longispinus”, Kurhade, Suresh E.; Siddaiah, V.; Bhuniya, Debnath; Reddy, D. Srinivasa, Synthesis, 2013, 45, 12, 1689-1692, DOI:10.1055/s-0033-1338450

“Synthesis of new binol based [1+1] macrocyclic chiral manganese(III) Schiff bases as catalysts for asymmetric epoxidation”, Suresh, Paulsamy; Srimurugan, Sankareswaran; Dere, Ravindra T.; Ragavan, R. Venkat; Gopinath, Vadiraj Suphala, Tetrahedron: Asymmetry, 2013,  24, 11, 669-676, DOI:10.1016/j.tetasy.2013.04.017

“Unprecedented N→C[1,4] Boc migration: synthesis of 3-carboxyl functionalized 7-azaindolo[2,1-c][1,4]benzoxazine ring system”, Kurhade, Santosh; Ramaiah, Parimi Atchuta; Prathipati, Philip; Bhuniya, Debnath, Tetrahedron, 2013, 69, 4, 1354-1362, DOI:10.1016/j.tet.2012.11.073

“Comparison of a High-Throughput High-Content Intracellular Leishmania donovani Assay with an Axenic Amastigote Assay”, Manu De Rycker, Irene Hallyburton, John Thomas, Lorna Campbell, Susan Wyllie, Dhananjay Joshi, Scott Cameron, Ian H. Gilbert, Paul G. Wyatt, Julie A. Frearson, Alan H. Fairlamb, David W. Gray. Antimicrobial Agents and Chemotherapy, 2013,
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“Acetamide compounds as glucokinase modulators and their preparation and use for treatment and prevention of glucokinase-mediated diseases”, Kurhade, Santosh; Kandalkar, Sachin; Kaduskar, Rahul; Kobal, Balasaheb; Naik, Keshav; Dave, Bhavesh; Deshpande, Anil; Bhuniya, Debnath; Palle, Venkata Poornapragnacharyulu, PCT Int. Appl., 2012, WO 2012020357 A1 20120216

“Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors”, Basu, Sujay; Prasad, Uppuleti Viplava; Barawkar, Dinesh A.; De, Siddhartha; Palle, Venkata P.; Menon, Suraj; Patel, Meena; Thorat, Sachin; Singh, Umesh P.; Sarma, Koushik Das; et al, Bioorganic & Medicinal Chemistry Letters, 2012, 22, 8, 2843-2849, DOI:10.1016/j.bmcl.2012.02.070

“Discovery of pyrazole carboxylic acids as potent inhibitors of rat long chain L-2-hydroxy acid oxidase”, Barawkar, Dinesh A.; Bandyopadhyay, Anish; Deshpande, Anil; Koul, Summon; Kandalkar, Sachin; Patil, Pradeep; Khose, Goraksha; Vyas, Samir; Mone, Mahesh; Bhosale, Shubhangi; et al, Bioorganic & Medicinal Chemistry Letters, 2012, 22, 13, 4341-4347, DOI:10.1016/j.bmcl.2012.05.020

“Inverse kinetic isotope effect in Magtrieve mediated oxidation or deoximation of benzaldoxime: mechanistic implication”, Bhosale, Sandeep; Sonune, Dnyaneshwar P.; Prasad, Uppuleti Viplava; Bhuniya, Debnath, Tetrahedron Letters,  2012, 53, 14, 1794-1797, DOI:10.1016/j.tetlet.2012.01.111

“Luseogliflozin: SGLT2 inhibitor treatment of diabetes”, Tiwari, A., Drugs of the Future, 2012, 37, 9, 637-643, DOI:10.1358/dof.2012.37.9.1848191

“Preparation of acetamide compounds as glucokinase activators, their process and medicinal applications”, Deshpande, Anil; Dave, Bhavesh; Kurhade, Santosh; Kobal, Balasaheb; Naik, Keshav; Kandalkar, Sachin; Bhuniya, Debnath; Palle, Venkata Poornapragnacharyulu, Eur. Pat. Appl., 2012, EP 2402327 A1 20120104

“Preparation of acetamide derivatives as glucokinase activators”, Bhuniya, Debnath; Bhosale, Sandeep Bhausaheb; De, Siddhartha; Palle, Venkata Poornapragnacharyulu, Indian Pat. Appl., 2012, IN 2007CH02266 A 20120921

“Preparation of acetamide derivatives as glucokinase activators”, Bhuniya, Debnath; Deshpande, Anil; Kandalkar, Sachin; Kobal, Balasaheb; Kurhade, Santosh; Vyavahare, Vinod; Kaduskar, Rahul, From U.S. Pat. Appl. Publ. (2012), US 20120214735 A1 20120823

“Preparation of fused pyrimidine compounds as therapeutic adenosine receptor antagonist”, Palle, Venkata; Basu, Sujay; Waman, Yogesh; Ramadas, Vidya; Barawkar, Dinesh, From Indian Pat. Appl., 2012, IN 2008CH00746 A 20120629

“Preparation of fused tricyclic compounds as therapeutic adenosine receptor antagonist”, Barawkar, Dinesh; Basu, Sujay; Ramdas, Vidya; Naykodi, Minakshi; Patel, Meena; Shejul, Yogesh; Thorat, Sachin; Panmand, Anil, PCT Int. Appl., 2012, WO 2012038980 A2 20120329

“Preparation of purine compounds as prodrugs of A2B adenosine receptor antagonists”, Barawkar, Dinesh; Basu, Sujay; Ramdas, Vidya; Palle, Venkata Poornapragnacharyulu; Waman, Yogesh; Patel, Meena; Panmand, Anil, Indian Pat. Appl., 2012, IN 2010CH02671 A 20120713

“Preparation of purine compounds as prodrugs of A2B adenosine receptor antagonists”, Barawkar, Dinesh; Basu, Sujay; Ramdas, Vidya; Palle, Venkata Poornapragnacharyulu; Waman, Yogesh; Patel, Meena; Panmand, Anil, PCT Int. Appl., 2012, WO 2012035548 A1 20120322

“Preparation of substituted fused pyrimidine compounds as adenosine receptor antagonists”,  Palle, Venkata; Ramdas, Vidya; Barawkar, Dinesh; Basu, Sujay; Koul, Summon; Waman, Yogesh, From Indian Pat. Appl., 2012, IN 2009CH00571 A 20120413

“Reevaluation of the Coding Potential and Proteomic Analysis of the BAC-Derived Rhesus Cytomegalovirus Strain 68-1”, Daniel Malouli, Ernesto S. Nakayasu, Kasinath Viswanathan, David G. Camp II, W. L. William Chang, Peter A. Barry, Richard D. Smith, Klaus Früh. American Society for Microbiology, 2012, DOI: 10.1128/JVI.01132-12.

“A Static-Cidal Assay for Trypanosoma brucei to Aid Hit Prioritisation for Progression into Drug Discovery Programmes”, Manu De Rycker, Sandra O’Neill, Dhananjay Joshi, Lorna Campbell, David W. Gray, Alan H. Fairlamb. PLOS Neglected Tropical Diseases, 2012, DOI: 10.1371/journal.pntd.0001932.

“Preparation of substituted fused tricyclic compounds as JAK kinase inhibitors, compositions and medicinal applications thereof”, Barawkar, Dinesh; Bende, Tanushree; Zahler, Robert; Bandyopadhyay, Anish; Sarangthem, Robindro Singh; Doshi, Jignesh; Waman, Yogesh; Jadhav, Rushikesh; Singh, Umesh Prasad, PCT Int. Appl., 2012, WO 2012127506 A1 20120927

“Substituted fused pyrimidine compounds, their preparation and therapeutic uses thereof”, Ramdas, Vidya; Koul, Summon; Basu, Sujay; Waman, Yogesh; Shejul, Yogesh; Barawkar, Dinesh; Palle, Venkata, Indian Pat. Appl., 2012, IN 2009CH02720 A 20120420

“A phosphine-mediated synthesis of 1,4-oxazepine- and 1,5-oxazocine-based sugar hybrids from deoxysugar azides”, Kurhade, Suresh E.; Salunkhe, Videsh T.; Siddaiah, V.; Bhuniya, Debnath; Reddy, D. Srinivasa, Synthesis, 2011, 21, 3523-3529, DOI:10.1055/s-0030-1260218

“An enantiospecific route to (+)-(1R,3S)-cis-chrysanthemic acid from (-)-D-pantolactone”, Hajare, Atul K.; Datrange, Laxmikant S.; Murthy, Y. L. N.; Bhuniya, Debnath; Reddy, D. Srinivasa, Synthesis, 2011, 7, 1067-1070, DOI:10.1055/s-0030-1258451

“Degradation Studies of Triprolidine: Isolation, Characterization of Oxidative Degradation Products and Development of A Validated Stability Indicating Uhplc Method”, Mone, Mahesh Kumar; Chandrasekhar, K. B.; Vyas, Samir, From Journal of Liquid Chromatography & Related Technologies, 2011, 34, 8, 652-669, DOI:10.1080/10826076.2011.558651

“Development of liquid chromatographic enantiomer separation methods and validation for the estimation of (R)-enantiomer in eslicarbazepine acetate”, Mone, Mahesh Kumar; Chandrasekhar, K. B., Journal of Pharmaceutical and Biomedical Analysis, 2011, 54, 1, 248-251, DOI:10.1016/j.jpba.2010.08.015

“Discovery of a potent and selective small molecule hGPR91 antagonist”, Bhuniya, Debnath; Umrani, Dhananjay; Dave, Bhavesh; Salunke, Deepak; Kukreja, Gagan; Gundu, Jayasagar; Naykodi, Minakshi; Shaikh, Nadim S.; Shitole, Prasad; Kurhade, Santosh; et al, Bioorganic & Medicinal Chemistry Letters,  2011, 21, 12, 3596-3602, DOI:10.1016/j.bmcl.2011.04.091

“Evaluation of Generic Gradients, Sample Pooling and MS Detection as Chiral Resolution Screening Strategies on Diverse Chiral Stationary Phases”, Mone, Mahesh Kumar; Chandrasekhar, K. B., Chromatographia, 2011, 73, 9-10, 985-992, DOI:10.1007/s10337-011-1980-z

“Fused nitrogen heterocyclic compounds as glucokinase modulators and their process for preparation and use in the treatment of glucokinase-mediated diseases”, Dave, Bhavesh; Deshpande, Anil; Kurhade, Santosh; Kobal, Balasaheb; Bhuniya, Debnath; Palle, Venkata, PCT Int. Appl., 2011, WO 2011080755 A1 20110707

“Potent and Selective Inhibitors of Long Chain L-2-Hydroxy Acid Oxidase Reduced Blood Pressure in DOCA Salt-Treated Rats”, Barawkar, Dinesh A.; Meru, Ashwin; Bandyopadhyay, Anish; Banerjee, Abir; Deshpande, Anil M.; Athare, Chandrashekhar; Koduru, Chandrasekhar; Khose, Goraksha; Gundu, Jayasagar; Mahajan, Koshu; et al, ACS Medicinal Chemistry Letters, 2011, 2, 12, 919-923, DOI:10.1021/ml2001938

“Preparation of benzamide compounds as glucokinase activators and their pharmaceutical application”,

Deshpande, Anil; Kandalkar, Sachin; Naik, Keshav; Dave, Bhavesh; Bhuniya, Debnath; Palle, Venkata, PCT Int. Appl., 2011, WO 2011095997 A1 20110811

“Regulated bioanalysis: an Indian perspective on harmonization efforts”, Ramanathan, Vikram K.; Vachharajani, Nimish N., Bioanalysis, 2011, 3, 7, 713-716, DOI:10.4155/bio.11.14

“Stereo-conserved synthesis of syn-diarylheptanoids, active principles of Zingiber, starting from D-glucose”, Bhosale, Sandeep; Vyavahare, Vinod P.; Prasad, Uppuleti Viplava; Palle, Venkata P.; Bhuniya, Debnath, Tetrahedron Letters, 2011, 52, 26, 3397-3400, DOI:10.1016/j.tetlet.2011.04.097

“Substituted fused pyrimidine compounds, its preparation and uses thereof”, Ramdas, Vidya; Koul, Summon; Basu, Sujay; Waman, Yogesh; Shejul, Yogesh; Barawkar, Dinesh; Palle, Venkata Poornapragnacharyulu, PCT Int. Appl., 2011, WO 2011055391 A1 20110512

“Synthesis and antimicrobial studies of some new 3-isoxazoline substituted phthalazine methylsulfonyl oxadiazoles”, Sridhara, A. M.; Venugopala Reddy, K. R.; Keshavayya, J.; Ambika, D. S.; Goud, Sanathkumar; Peethambar, S. K., E-Journal of Chemistry, 2011, 8, 3, 1022-1029, DOI:10.1155/2011/356437

“International recommendations for training future toxicologic pathologists participating in regulatory-type, nonclinical toxicity studies☆”, Brad Bolona, Erio Barale-Thomas, Alys Bradley, Robert A. Ettlin, Carla A. S. Franchi, Catherine George, Anna Maria Giusti, Robert Hall, Matthew Jacobsen, Yoichi Konishi, David Ledieu, Daniel Morton, Jae-Hak Park, Cheryl L. Scudamore, Hiroyuki Tsuda, S. K. Vijayasarathi, Marcel V. W. Wijnands. Experimental and Toxicologic Pathology, 2011, 63(1-2), 187-195, DOI: 10.1016/j.etp.2010.07.006.

“Validation of 96-well Equilibrium Dialysis with Non-radiolabeled Drug for Definitive Measurement of Protein Binding and Application to Clinical Development of Highly-Bound Drugs”, Maciej J. Zamek-Gliszczynski, Kenneth J. Ruterbories, Rose T. Ajamie, Enaksha R. Wickremsinhe, Lavanya Pothuri, Mukkavilli V. S. Rao, Vinay N. Basavanakatti, Jakir Pinjari, Vikram K. Ramanathan, Ajai K. Chaudhary. Journal of Pharmaceutical Sciences, 2011, 100(6), 2498-2507, DOI: 10.1002/jps.22452

“Synthesis of a novel tetracyclic azaindolo[2,1-c][1,4]benzoxazine ring system”, Kurhade, Santosh; Kaduskar, Rahul D.; Dave, Bhavesh; Ramaiah, Parimi Atchuta; Palle, Venkata P.; Bhuniya, Debnath, Tetrahedron Letters, 2011, 52, 16, 1874-1877, DOI:10.1016/j.tetlet.2011.02.020

“Synthesis of Molluscicidal Agent Cyanolide A Macrolactone from D-(-)-Pantolactone”, Hajare, Atul K.; Ravikumar, Velayutham; Khaleel, Shaik; Bhuniya, Debnath; Reddy, D. Srinivasa, Journal of Organic Chemistry, 2011, 76, 3, 963-966, DOI:10.1021/jo101782q

“Synthesis of novel dihydrooxazine and oxazoline based sugar hybrids from sugar azides”, Kurhade, Suresh E.; Ravula, Sudhir; Siddaiah, V.; Bhuniya, Debnath; Reddy, D. Srinivasa, Tetrahedron Letters, 2011, 52, 33, 4313-4315, DOI:10.1016/j.tetlet.2011.06.035

“Synthesis of novel sugar-lactam conjugates using the Aube reaction”, Kurhade, Suresh E.; Mengawade, Tanaji; Bhuniya, Debnath; Palle, Venkata P.; Reddy, D. Srinivasa, Organic & Biomolecular Chemistry, 2011, 9, 3, 744-747, DOI:10.1039/C0OB00719F

“Synthesis, antimicrobial and cytotoxicity studies of some novel modified strobilurin derivatives”, Sridhara, Ajjanna M.; Reddy, Kallam R. Venugopala; Keshavayya, Jathi; Ambika, Dasannana Malige S.; Gopinath, Vadiraj S.; Bose, Prosenjit; Goud, Sanath Kumar; Peethambar, Sanenahalli K., Journal of the Brazilian Chemical Society, 2011, 22, 5, 849-856, DOI:10.1590/S0103-50532011000500006

“Synthesis, antimicrobial and cytotoxicity studies of some novel phthalazine-methoxyacrylate derivatives”, Sridhara, Ajjanna M.; Reddy, Kallam R. Venugopala; Keshavayya, Jathi; Vadiraj, Suphala G.; Bose, Prosenjit; Ambika, D. S.; Raju, Ch. Krishnam; Shashidhara, S.; Raju, N. Hanumantha, Journal of Pharmacy Research, 2011, 4, 2, 496-500

“Total Synthesis of Isofregenedadiol”, Kurhade, Suresh E.; Sanchawala, Abbas I.; Ravikumar, Velayutham; Bhuniya, Debnath; Reddy, D. Srinivasa, Organic Letters, 2011, 13, 14, 3690-3693, DOI:10.1021/ol201336x

“Degradation studies of pentoxifylline: Isolation and characterization of a novel gem-dihydroperoxide derivative as major oxidative degradation product”, Mone, Mahesh Kumar; Chandrasekhar, K. B., Journal of Pharmaceutical and Biomedical Analysis, 2010, 53, 3, 335-342, DOI:10.1016/j.jpba.2010.04.006

“Direct nuclear halogenation of deactivated aryl and N-heteroaryl amines”, Waghmare, Anirudha A.; Bose, Prosenjit; Pati, Hari N., Pharma Chemica, 2010, 2, 5, 212-241

“Enantiospecific synthesis of sex pheromone of the obscure mealybug from pantolactone via tandem conjugate addition/cyclization”, Hajare, Atul K.; Datrange, Laxmikant S.; Vyas, Samir; Bhuniya, Debnath; Reddy, D. Srinivasa, Tetrahedron Letters, 2010, 51, 40, 5291-5293, DOI:10.1016/j.tetlet.2010.07.166

“Magtrieve (CrO2) and MnO2 mediated oxidation of aldoximes: studying the reaction course”, Bhosale, Sandeep; Kurhade, Santosh; Vyas, Samir; Palle, Venkata P.; Bhuniya, Debnath, Tetrahedron, 2010, 66, 50, 9582-9588, DOI:10.1016/j.tet.2010.10.029

“Preparation of acetamide derivatives as glucokinase activators”, Bhuniya, Debanath; Bhosale, Sandeep Bhausaheb; Kapkoti, Gobind Sing; Palle, Venkata Poornapragnacharyulu; De, Siddhartha; Mookhtiar, Kasim A.; Dave, Bhavesh; Deshpande, Anil; Kurhade, Santosh; Kobal, Balasaheb; et al, U.S. Pat. Appl. Publ. (2010), US 20100310493 A1 20101209

“Protein binding in drug discovery and development”,  Ramanathan, Vikram; Vachharajani, Nimish Edited By:Han, Chao; Davis, Charles B.; Wang, Binghe, Evaluation of Drug Candidates for Preclinical Development, 2010, 135-167, DOI:10.1002/9780470574898.ch6

“Substituted fused pyrimidine compounds”, Palle, Venkata; Ramdas, Vidya; Barawkar, Dinesh; Basu, Sujay; Koul, Summon; Waman, Yogesh; Patel, Meena; Panmand, Anil, PCT Int. Appl., 2010, WO 2010103547 A2 20100916

“Synthesis and antimicrobial activity of 2-substituted [4-(1,3,4-oxadiazol-2-yl methyl)]phthalazin-1(2H)-one derivatives”, Sridhara, Ajjanna M.; Venugopala Reddy, Kallam R.; Keshavayya, Jathi; Kumar Goud, Palusa Sanath; Somashekar, Bankavadi C.; Bose, Prosenjit; Peethambar, Sanenahalli K.; Gaddam, Satish Kumar, European Journal of Medicinal Chemistry,  2010, 45, 11, 4983-4989, DOI:10.1016/j.ejmech.2010.08.005

“Synthesis and antimicrobial activity of phthalazine substituted 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazoles and 7H-[1,2,4]triazolo[3,4-b]thiadiazines”, Sridhara, A. M.; Reddy, K. R. Venugopala; Keshavayya, J.; Chidananda, B.; Prasad, Yaragola; Kumar, G. Satish; Vadiraj, S. G.; Bose, Prosenjit; Goud, Sanath Kumar; Peethambar, S. K., Pharma Chemica, 2010, 2, 5, 201-211

“Titrimetric assay of lisinopril in aqueous and non-aqueous media”, K. Basavaiah, K. Tharpa, K. B. Vinay. Ecletica Quimica Journal, 2010, 35(2), DOI: 10.26850/1678-4618eqj.v35.2.2010.p07-14.

“Is contract broiler farming exploitative to small farmers?”, R. K. Thamizhselvi, S. V. N. Rao. The Indian journal of animal sciences, 2010, 80(12), 1243-1250

“Sensitive spectrophotometric assay of simvastatin in pharmaceuticals using permanganate”, Kalsang Tharpa, Kanakapura Basavaiah, Nagaraju Rajedraprasad, Kanakapura Basavaiah Vinay, Salmara Ganeshbhat Hiriyanna. Brazilian Journal of Pharmaceutical Sciences, 2010, 46(1), DOI: 10.1590/S1984-82502010000100010.

“Characterization of active and inactive states of CB1 receptor and the differential binding state modulation by cannabinoid agonists, antagonists and inverse agonists”, Srinivas Gullapalli, Dipak Amrutkar, Sangeetha Gupta, Machender R. Kandadi, Hemant Kumar, Maulik Gandhi, Vikas Karande, Shridhar Narayanan. Neuropharmacology, 2010, 58(8), 1215-1219, DOI: 10.1016/j.neuropharm.2010.03.001.

“Acute toxic effects of Endosulfan 35 EC (Endocel) upon oral gavage and dietary admixture in Japanese quails”, Prakash, P. J.; Rajashekhar, G.; Krishnappa, H.; Sulaiman, S. M.; Rao, K. Venugopala, Research Journal of Environmental Toxicology, 2009, 3, 3, 124-131, DOI:10.3923/rjet.2009.124.131

“Effect of Endosulfan 35% EC on the egg laying and egg shell thickness in Japanese quails”, Prakash, P. J.; Rajashekhar, Geetha; Krishnappa, H.; Sulaiman, S. M.; Venugopala Rao, K., Research Journal of Environmental Toxicology, 2009, 3, 3, 140-146, DOI:10.3923/rjet.2009.140.146

“Efficient synthesis of isoxazoles and isoxazolines from aldoximes using Magtrieve (CrO2)”, Bhosale, Sandeep; Kurhade, Santosh; Prasad, Uppuleti Viplava; Palle, Venkata P.; Bhuniya, Debnath, Tetrahedron Letters, 2009, 50, 27, 3948-3951, DOI:10.1016/j.tetlet.2009.04.073

“Preparation of acetamide derivatives as glucokinase activators”, Bhuniya, Debanath; Bhosale, Sandeep Bhausaheb; Kapkoti, Gobind Sing; Palle, Venkata Poornapragnacharyulu; De, Siddhartha; Mookhtiar, Kasim A., PCT Int. Appl., 2009, WO 2009047798 A2 20090416

“Preparation of pyrimidine compounds as therapeutic adenosine receptor antagonist”, Palle, Venkata; Basu, Sujay; Waman, Yogesh; Ramdas, Vidya; Barawkar, Dinesh, PCT Int. Appl., 2009, WO 2009118759 A2 20091001

“Titrimetric and Spectrophotometric Assay of Pantoprazole in Pharmaceuticals Using Permanganate”, Kanakapura Basavaiah, Nagaraju Rajendraprasad, Kalsang Tharpa, Urdigere Rangachar Anilkumar, Salamara Ganeshbhat Hiriyanna, Kanakapura Basavaiah Vinay. Journal of the Mexican Chemical Society, 2009, 53(1).

“Determination of raloxifene hydrochloride in human urine by LC-MS-MS”, Kumar Anil Urdigere R., Basavaiah Kanakapura, Tharpa Kalsang, Vinay Kanakapura B. Chemical Industry and Chemical Engineering Quarterly, 2009, 15(3), 119-123, DOI: 10.2298/CICEQ0903119K.

“A convenient and practical synthesis of Olmesartan medoxomil methyl ether”, Pati, Hari Narayan; Lahiri, Saswata; Sabbam, Ramesh Kumar; Vangala, Vijaya Bhaskar; Ramalingam, Boobalan; Hiriyanna, Salmara Ganeshbhat; Bose, Prosenjit,  Journal of Heterocyclic Chemistry, 2008, 45, 3, 917-920, DOI:10.1002/jhet.5570450342

“Acridones circumvent P-glycoprotein-associated multidrug resistance (MDR) in cancer cells”, Gopinath, Vadiraj S.; Thimmaiah, Padma; Thimmaiah, Kuntebommanahalli N., Bioorganic & Medicinal Chemistry, 2008, 16, 1, 474-487, DOI:10.1016/j.bmc.2007.09.020

“Preparation of phenoxythiazolylalkylacetamide derivatives and analogs as glucokinase activators”, Mookhtiar, Kasim A.; Bhuniya, Debnath; Dave, Bhavesh; Kapkoti, Gobind S.; Basu, Sujay; Chugh, Anita; De, Siddartha; Palle, Venkata P., PCT Int. Appl., 2008, WO 2008104994 A2 20080904

“Preparation of pyrrole-2-carboxamide derivatives as glucokinase activators and their pharmaceutical application”, Bhuniya, Debnath; Kapkoti, S. Gobind; Warrier, S. Jayakumar; Kukrejka, Gagan; Mavinahalli, N. Jagadeesh; Palle, P. Venkata; Mookhtiar, A. Kasim, PCT Int. Appl., 2008, WO 2008149382 A1

“Simultaneous determination of several angiotensin-II receptor antagonists by liquid chromatography”, Hiriyanna, S. G.; Basavaiah, K.; Dhayanithi, V.; Bindu, A.; Pujari, Sudhaker; Pati, Hari N., Analytical Chemistry: An Indian Journal, 2008, 7, 8, 568-572

“Unusual detritylation of tritylated tetrazole in sartan molecules”, Srimurugan, Sankareswaran; Suresh, Paulsamy; Babu, Balaji; Hiriyanna, Salmara Ganeshbhat; Pati, Hari Narayan, Chemical & Pharmaceutical Bulletin, 2008, 56, 3, 383-384, DOI:10.1248/cpb.56.383

“Uptake and persistence of soil applied paclobutrazol in ‘Alphonso’ mango and soil in the Konkan region of Maharashtra, India”, Debi Sharma, L. Shalini, M. Edward Raja. Toxicological & Environmental Chemistry, 2008, 90(3), 577-583, DOI: 10.1080/02772240701609756.

“Validated spectrophotometric methods for the determination of raloxifene hydrochloride in pharmaceuticals”, K Basavaiah, U R Anil Kumar, Kalsang Tharpa, K B Vinay. Journal of the Chilean Chemical Society, 2008, 1635-1639, DOI: 10.4067/S0717-97072008000300020.

“A facile synthesis of new chiral [1+1] macrocyclic schiff bases”, Suresh, Paulsamy; Srimurugan, Sankareswaran; Pati, Hari N., Chemistry Letters,  2007, 36, 11, 1332-1333, DOI:10.1246/cl.2007.1332

“Isolation by preparative HPLC and characterization of process-related impurities in tebuconazole”, Hiriyanna, S. G.; Sreedhar, K.; Dhayanithi, V.; Reddy, K. V. S. R. Krishna; Vaidyanathan, Gopal; Basavaiah, K., Analytical Chemistry: An Indian Journal, 2007, 5, 1-6, 51-56

“Microwave-assisted synthesis of 72-membered chiral hexanuclear [6 + 6] macrocyclic Schiff base”, Srimurugan, Sankareswaran; Suresh, Paulsamy; Pati, Hari N., Journal of Inclusion Phenomena and Macrocyclic Chemistry, 2007, 59, 3-4, 383-388, DOI:10.1007/s10847-007-9341-0

“Pharmacological and X-Ray Structural Characterization of a Novel Selective Androgen Receptor Modulator: Potent Hyperanabolic Stimulation of Skeletal Muscle with Hypostimulation of Prostate in Rats”, Jacek Ostrowski, Joyce E. Kuhns, John A. Lupisella, Mark C. Manfredi, Blake C. Beehler, Stanley R. Krystek, Jr., Yingzhi Bi, Chongqing Sun, Ramakrishna Seethala, Rajasree Golla, Paul G. Sleph, Aberra Fura, Yongmi An, Kevin F. Kish, John S. Sack, Kasim A. Mookhtiar, Gary J. Grover, Lawrence G. Hamann. Endocrinology, 2007, 148(1), 4–12, DOI: 10.1210/en.2006-0843.

“A rapid, homogeneous, fluorescence polarization binding assay for peroxisome proliferator-activated receptors alpha and gamma using a fluorescein-tagged dual PPARα/γ activator”, Ramakrishna Seethala, Rajasree Golla, Zhengping Ma, Hao Zhang, Kevin O’Malley, Jonathan Lippy, Lin Cheng, Kasim Mookhtiar, Dennis Farrelly, Litao Zhang, Narayanan Hariharan, Peter T.W.Cheng. Analytical Biochemistry, 2007, 363(2), 263-274, DOI: 10.1016/j.ab.2007.01.022.

“Modulation of metabolic enzymes by dietary phytochemicals: a review of mechanisms underlying beneficial versus unfavorable effects”, Mandlekar Sandhya; Hong Jin-Liern; Kong Ah-Ng Tony, Current drug metabolism, 2006, 7, 6, 661-75

“Muraglitazar, a Novel Dual (α/γ) Peroxisome Proliferator–Activated Receptor Activator, Improves Diabetes and Other Metabolic Abnormalities and Preserves β-Cell Function in db/db Mice”, Thomas Harrity, Dennis Farrelly, Aaron Tieman, Cuixia Chu, Lori Kunselman, Liqun Gu, Randolph Ponticiello, Michael Cap, Fucheng Qu, Chunning Shao, Wei Wang, Hao Zhang, William Fenderson, Sean Chen, Pratik Devasthale, Yoon Jeon, Ramakrishna Seethala, Wen-Pin Yang, Jimmy Ren, Min Zhou, Denis Ryono, Scott Biller, Kasim A. Mookhtiar, John Wetterau, Richard Gregg, Peter T. Cheng, Narayanan Hariharan. American Diabetes Association, 2006, 55(1), 240-248, DOI: 10.2337/diabetes.55.01.06.db05-0648.

Posters/Presentations

“Comparative Toxicity of Dimethoate to Honeybees, Apis cerena and Apis mellifera”, KP, Raveesha; Halappa, Ramesh; RS, Gangadhar; H, Mahesh; GC, Sunil; and V., Pardhasaradhi., 2020, SETACSciCon (SETAC Europe 30th Annual Meeting), Poster ID:2.02P.6

“In vitro Metabolism and Disposition of DNDI-VL-2098, a Potential Treatment for Visceral Leishmaniasis”, Rao, MVS; Pinjari, Jakir; Pothuri, Lavanya; Mondal, Subodh; Gopu, C.L.; Prabhakar, K.R.; Launay, Delphine; Martin, Denis; Vachharajani, Nimish; Ramanathan, Vikram., 2011, AAPS, Poster No: R6388

“Preclinical Pharmacokinetics and Prediction of Human PK of DNDI-VL-2098, a Potential Oral Treatment for Visceral Leishmaniasis”, Harisudhan, T.; Pinjari, Jakir; Gadekar, Ajit; Verma, Manas; Patel, Bhavesh; Patel, Jignesh; Moinuddin, F.; Shankar, S.; Rao, MVS; Launay, Delphine; Martin, Denis; Vachharajani, Nimish; Ramanathan, Vikram., 2011, AAPS, Poster No: R6389

“Buparvaquone Pharmacokinetics and its Solubility-Limited Oral Absorption”, Pinjari, Jakir; Badrinath, R; Jayasagar, G; Kanchi, R; Nageswararao, K; Pasha, Mazhar; Rohith, N; Vinay, H Vachharajani, Nimish; Ramanathan, Vikram.,AAPS, 2008, Poster No: M1305

“Hydroxychloroquine Pharmacokinetics and Tissue Distribution in the C57 black mouse”, Raff, Howard; Jayasagar, G; Bhatt, Deepak; Nigade, Prashant; Pinjari, Jakir; Rao, Mukkavilli; Shankar, S; Sivaprasad, Putlur; Vachharajani, Nimish; Ramanathan, Vikram., 2008, AAPS, Poster No: M1315